All you need to know about preparations with the active substance Anastrozole

Anastrozole is an active substance that has found wide application in medicine and sports pharmacology. It belongs to a group of drugs known as aromatase inhibitors. Aromatase is an enzyme responsible for converting male hormones (such as testosterone) into female hormones (estrogens). Anastrozole inhibits the activity of aromatase, resulting in lower oestrogen levels.

Anastrozole is also used by men to achieve the same effect – lowering estrogen levels. This is especially true in the context of bodybuilding and anabolic steroid use. Estradiol is one of the main estrogens, which is formed from testosterone with the help of aromatase. The use of anastrozole in men reduces the conversion of testosterone to estrogens by inhibiting aromatase activity.

Thus, in bodybuilding and sports circles, anastrozole-based drugs are widely used to prevent or reduce unwanted estrogenic side effects associated with the use of anabolic steroids. These may include gynaecomastia, fluid retention and other adverse effects associated with estrogenic activity.

  • The ATX (Anatomical-Therapeutic-Chemical Classification) code for anastrozole is L02BG03. This is a code used to classify drugs according to their pharmacological and therapeutic properties.
  • Structural formula of anastrozole: C17H19N5.
  • Clinical and pharmacological group: Hormone antagonists and related agents. Aromatase inhibitors. Antitumour preparations

Anastrozole manufacturer prices may vary depending on the dosage form, brand, country of production and sale of the remedy, concentration of the mixture and other factors.

Advantages and effects of drugs

Medicines containing the active ingredient anastrozole have several effects that have made them popular in bodybuilding:

  • Reduction of oestrogen levels. The main mechanism of action is inhibiting the activity of aromatase, the enzyme responsible for converting testosterone into estrogens. This reduces oestrogen levels in the body, which can be beneficial in a variety of clinical and athletic situations.
  • Reducing the risk of breast cancer. Anastrozole can also be used to reduce the risk of developing breast cancer. For women at increased risk of developing breast cancer, anastrozole may be an effective preventative treatment.
  • Preventing side effects of anabolic steroids. In bodybuilders using anabolic steroids, anastrozole may be effective in reducing unwanted estrogenic side effects such as gynaecomastia, fluid retention and fat retention.
  • Improving symptoms of hyperestrogenism. Some men and women who are undergoing a course of lean and/or muscle building may experience elevated levels of oestrogen in the body, with associated symptoms. Anastrozole helps to improve the symptoms of hyperestrogenism (hormonal imbalances, skin problems, etc.).

Preparations of the active ingredient anastrozole in bodybuilding have many advantages. Bodybuilders prefer to buy anastrozole, particularly for SCT, because it has no progestagenic, estrogenic and androgenic activity. As our tests have shown, these drugs in therapeutic doses of the substance also have no effect on the secretion of aldosterone and cortisol in the body.

Scientific substantiation and clinical studies of Anastrozole

Anastrozole was subjected to clinical trials, which allowed us to identify its potential side effects and interactions with other drugs. We have relied on their results, comparing them with our own experience:

  • The ATAC study. This compared the effects of anastrozole and tamoxifen in the treatment of breast cancer in postmenopausal women. The results showed that anastrozole was more effective than tamoxifen in reducing the risk of breast cancer recurrence.
  • IBIS-II study. A course of Anastrozole was used to reduce the risk of breast cancer. The results showed that Anastrozole significantly reduced the risk of breast cancer in at-risk female patients.
  • Study MA.27: Anastrozole was used as maintenance therapy after primary treatment for breast cancer in postmenopausal women. Results showed that the drug reduced the risk of recurrence and improved survival in female patients.
  • Studies were conducted on men to examine the effects of anastrozole on reducing oestrogen levels and improving symptoms of hyperestrogenism associated with anabolic steroid use. Anastrozole was effective.

The studies provided a scientific basis for the use of anastrozole and confirmed its safety and good tolerability. Once we tested it in practice, we were able to evaluate its efficacy and safety in a variety of conditions personally. Anastrozole has proven to be really effective in lowering oestrogen levels and preventing the side effects associated with the use of anabolic steroids. It is excreted from the body naturally. After taking 1 dose of the drug, the excretion process is up to 72 h.

Guidelines for dosage and cycles of administration of preparations with the active substance Anastrozole

Usually the recommended dose of anastrozole is 1 mg per day, and the course lasts 20-28 days, so the price for anastrozole is usually indicated for 20-28 tablets of exactly this dosage. However, it can be adjusted by a doctor depending on individual factors. Based on our observations, the optimal dosage for reducing estrogenic side effects associated with anabolic steroid use would be 0.5 mg-1 mg per day.

Specific guidance on cycles of use requires medical judgement and individualisation. The dosage and regimen may vary depending on the patient’s specific medical condition, treatment goals, and other factors. Improper use can lead to unwanted side effects and complications. That is why you can buy anastrozole in the United Kingdom without a prescription only from online shops – pharmacies will require a doctor’s recommendation.

We recommend that you speak to your doctor or pharmacist. Only they can advise according to your individual needs, which will help to avoid overdose.

Safety and side effects 

Anastrozole is well tolerated by patients, but as with any medication, side effects can occur:

  • Headache may occur in some patients.
  • Some patients may experience muscle and/or joint pain.
  • Hypercholesterolaemia: Anastrozole may increase blood cholesterol levels.
  • Postmenopausal women may have an increased risk of osteoporosis (worsening bone density).
  • Some studies suggest that anastrozole may be associated with an increased risk of cardiovascular disease, such as myocardial infarction and stroke.
  • Some patients may experience sleep problems or sleep disturbances.
  • The strain on the liver that any pill places on the liver prevents it from being taken by people suffering from diseases of this organ.

If you experience any side effects while taking anastrozole, it is important to see a doctor who will assess their severity and decide on further treatment. The doctor can decide to adjust the dose and minimise side effects, tell you how to take anastrozole in bodybuilding on a drying course or SCT.

Indications for the use of preparations with the active substance Anastrozole

Anastrozole is sometimes used in bodybuilding to lower oestrogen levels and prevent unwanted estrogenic side effects associated with the use of anabolic steroids. Some indications for a course of Anastrozole supplementation for bodybuilders, include:

  • Lowering oestrogen levels. Anastrozole can help lower oestrogen levels in a bodybuilder’s body, especially when using anabolic steroids, which can cause oestrogen levels to rise.
  • Side Effect Control. Anastrozole can help control and prevent the development of side effects associated with anabolic steroid use, such as water retention, high blood pressure, and gynaecomastia.
  • Improved physical fitness. By lowering oestrogen levels, anastrozole can help improve a bodybuilder’s fitness, allowing them to achieve leaner and more beautiful looking muscles.

Remember: the use of anastrozole in bodybuilding should be supervised by a doctor. It is necessary to follow the recommendations of a specialist regarding the dosage and regimen to avoid unwanted side effects.

Opinions of users about drugs with the active substance Anastrozole

Opinions about the drugs turned out to be diverse. This is not surprising – each person is different. Some noted positive effects and good tolerance of the drugs, others had side effects – muscle and joint pain, headache, sleep disturbance and depression. A few users, according to them, did not achieve the expected results.

But in general, reviews of women taking anastrozole, as well as male athletes, confirm its effectiveness:

  • Many noted a decrease in oestrogen levels, which helped them achieve leaner fitness and avoid the unwanted effects associated with high oestrogen levels.
  • Anastrozole has been effective in preventing gynaecomastia.
  • Some have noted an improvement in their overall condition, increased energy and decreased fatigue.

Everyone may have a different individual reaction, effectiveness and tolerability will vary. It is important to realise that users’ opinions are based on their own experiences and they may vary. For some, the disadvantage was how much does anastrozole cost, while others, after comparing prices in different countries, found it quite cheap compared to its analogues.

Where to buy Anastrozole in the United Kingdom: reliable suppliers

You can buy Anastrozole in the United Kingdom in a regular pharmacy or online. If you choose the first option, you should take care to get a prescription from your doctor. In the second case, you will not need to do this, but it is important to choose a reliable supplier. Make sure that the product is original.

At Anastrozolebodybuilding shop, where you can buy anastrozole at manufacturer’s prices, anonymously and without a prescription, you will find products with anti-counterfeit labelling. We provide optimal conditions of delivery and storage of funds to extend their life.

By choosing our shop, you start a cooperation with responsible specialists, and you can count on the highest quality of pharmaceutical products that can only be found on this market. Contact a consultant to get answers to your questions. You can place your order through the shopping basket – just fill in the feedback form.

Most frequently asked questions about preparations with the active substance Anastrozole

1.Does Anastrozole reduce libido?

– If taken correctly, this should not happen. Anastrozole is neutral for potency. If you notice a worsening of potency after taking Anastrozole, try lowering the dosage.

2.What drug can be substituted for Anastrozole?

– Possible alternatives to Anastrozole may include other aromatase inhibitors such as letrozole or exemestane. Substitution can only be discussed with a medical professional, as the choice of an alternative drug depends on the specific situation, individual patient characteristics and treatment goals. 

3.How much does anastrozole reduce estradiol levels?

– In women, when taking 1 mg per day, there is a decrease in the concentration of estradiol up to 80%. In men, on the other hand, this drug usually causes a decrease in estradiol levels of about 50%.

4.Is it allowed to take Anastrozole before competition?

– Some organisations may prohibit the use of Anastrozole. It is important to check the official regulations of the organiser to find out for sure.

5.Can I buy Anastrozole anonymously?

– Yes, from online shops. You will need a prescription from a doctor to buy from a pharmacy.

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