Description
Anastrozol is an “anti-aromatase” tablet drug used by many bodybuilders to prevent gynecomastia and edema – side effects associated with the use of testosterone esters. Anastrozole is the most popular, guaranteed fastest way to get rid of aromatization and its effects in the early stages. It works much more effectively than other well-known anti-aromatase drugs such as Tamoxifen or Nolvadex.
Aromatase is a key enzyme in estrogen biosynthesis.
Anastrozole reduces aromatase activity by about 95% of the baseline level.
Anastrozole has a specific inhibitory effect on aromatase, unlike megestrol acetate or aminoglutethimide.Anastrozole does not affect adrenal steroidogenesis.
Anastrozole is able to inhibit aromatization highly effectively. The drug is rapidly and completely absorbed from the gastrointestinal tract, the maximum concentration of the drug in the blood is reached 2 h after ingestion on an empty stomach, metabolized slowly and, therefore, has a relatively long half-life (40-50 h), excreted mainly with urine and in smaller amounts – with bile.
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